Eg5 Inhibitor V, trans-24
CAS No. 869304-55-2
Eg5 Inhibitor V, trans-24( —— )
Catalog No. M26190 CAS No. 869304-55-2
Eg5 Inhibitor V, trans-24 is a specific and potent Eg5 agonist inhibitor that can be used in cancer research with an IC50 value of 0.65 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 227 | In Stock |
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| 5MG | 204 | In Stock |
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| 10MG | 306 | In Stock |
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| 25MG | 494 | In Stock |
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| 50MG | 663 | In Stock |
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| 100MG | 886 | In Stock |
|
| 200MG | 1190 | In Stock |
|
| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameEg5 Inhibitor V, trans-24
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NoteResearch use only, not for human use.
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Brief DescriptionEg5 Inhibitor V, trans-24 is a specific and potent Eg5 agonist inhibitor that can be used in cancer research with an IC50 value of 0.65 uM.
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DescriptionEg5 Inhibitor V, trans-24 is a specific and potent Eg5 agonist inhibitor that can be used in cancer research with an IC50 value of 0.65 uM.(In Vitro):Trans-24 is a potent EG5-specific inhibitor with an IC50 conversion rate of 0.65 M and can be used in cancer research.
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In VitroEg5 Inhibitor V, trans-24 is a potent and specific Eg5 inhibitor with an IC50 of 0.65 μM, and can be used in the research of cancer.
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In Vivo——
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Synonyms——
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PathwayCytoskeleton/Cell Adhesion Molecules
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TargetKinesin
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RecptorDyrk pS421| Dyrk1B
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Research Area——
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Indication——
Chemical Information
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CAS Number869304-55-2
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Formula Weight423.472
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Molecular FormulaC26H21N3O3
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Purity>98% (HPLC)
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Solubility——
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SMILES[H][C@@]12Cc3c([nH]c4ccccc34)[C@H](N1C(=O)N(Cc1ccccc1)C2=O)c1cccc(O)c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Kettle JG, et al. Discovery and optimization of a novel series of Dyrk1B kinase inhibitors to explore a MEK resistance hypothesis. J Med Chem. 2015 Mar 26;58(6):2834-44.
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