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Takeda103A
CAS No. 865609-72-9
Takeda103A( Takeda-103-A | Takeda 103 A | Takeda-103A | CMPD103A | CMPD-103A )
Catalog No. M24868 CAS No. 865609-72-9
Takeda103A is the GRK2-dependent bovine tubulin oxidation effective inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 186 | In Stock |
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| 2MG | 102 | In Stock |
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| 5MG | 159 | In Stock |
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| 10MG | 257 | In Stock |
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| 25MG | 424 | In Stock |
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| 50MG | 551 | In Stock |
|
| 100MG | 770 | In Stock |
|
| 200MG | 1014 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTakeda103A
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NoteResearch use only, not for human use.
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Brief DescriptionTakeda103A is the GRK2-dependent bovine tubulin oxidation effective inhibitor.
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DescriptionTakeda103A is the GRK2-dependent bovine tubulin oxidation effective inhibitor.
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In Vitro——
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In Vivo——
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SynonymsTakeda-103-A | Takeda 103 A | Takeda-103A | CMPD103A | CMPD-103A
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PathwayOthers
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TargetGRK (GPCRK)
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RecptorGRK2
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Research Area——
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Indication——
Chemical Information
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CAS Number865609-72-9
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Formula Weight463.49
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Molecular FormulaC24H23F2N7O
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Purity>98% (HPLC)
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SolubilityDMSO:10 mM
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SMILESCCCN1C(=NN=C1C2=NC=NC=C2)CNC3=CC=CC(=C3)C(=O)NCC4=C(C=CC=C4F)F
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Waldschmidt HV, Homan KT, Cruz-Rodríguez O, et al. Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors. J Med Chem. 2016 Apr 28;59(8):3793-807. doi: 10.1021/acs.jmedchem.5b02000. Epub 2016 Apr 13. PubMed PMID: 27050625.
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