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CB1 antagonist 2
CAS No. 614726-85-1
CB1 antagonist 2( AM4113 )
Catalog No. M24614 CAS No. 614726-85-1
CB1 antagonist 2 is caimabinoid 1 (CB1) antagonist extracted from patent WO2016184310A1, compound 3. Which inhibits CB1 in vivo with an IC50 of 25.5 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 29 | In Stock |
|
| 5MG | 42 | In Stock |
|
| 10MG | 69 | In Stock |
|
| 25MG | 141 | In Stock |
|
| 50MG | 245 | In Stock |
|
| 100MG | 398 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 900 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCB1 antagonist 2
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NoteResearch use only, not for human use.
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Brief DescriptionCB1 antagonist 2 is caimabinoid 1 (CB1) antagonist extracted from patent WO2016184310A1, compound 3. Which inhibits CB1 in vivo with an IC50 of 25.5 nM.
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DescriptionCB1 antagonist 2 is caimabinoid 1 (CB1) antagonist extracted from patent WO2016184310A1, compound 3. Which inhibits CB1 in vivo with an IC50 of 25.5 nM.
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In Vitro——
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In Vivo——
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SynonymsAM4113
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PathwayGPCR/G Protein
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TargetCannabinoid Receptor
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RecptorCB1
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Research Area——
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Indication——
Chemical Information
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CAS Number614726-85-1
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Formula Weight380.66
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Molecular FormulaC17H12Cl3N3O
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Purity>98% (HPLC)
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SolubilityDMSO: 60 mg/mL (157.62 mM; Need ultrasonic); H2O: < 0.1 mg/mL (insoluble)
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SMILESCc1c(-c(cc2)ccc2Cl)n(-c(ccc(Cl)c2)c2Cl)nc1C(N)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Li, S. , et al. "4-methyl-1h-diaryl pyrazole derivatives and their uses as medicament." WO, WO2007121687 A1.
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