AZD5305

CAS No. 2589531-76-8

AZD5305( —— )

Catalog No. M24160 CAS No. 2589531-76-8

AZD5305 is a potent, selective and oral active PARP inhibitor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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10MG 357 In Stock
25MG 597 In Stock
50MG 851 In Stock
100MG 1152 In Stock
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Biological Information

  • Product Name
    AZD5305
  • Note
    Research use only, not for human use.
  • Brief Description
    AZD5305 is a potent, selective and oral active PARP inhibitor.
  • Description
    AZD5305 is a potent, selective and oral active PARP inhibitor.
  • In Vitro
    ——
  • In Vivo
    Animal Model:Female Han Wistar rats with BRCAm xenograft and PDX models (12-13 weeks of age)Dosage:0.01, 0.03, 0.1, and 0.3 mg/kg Administration:Oral administration; daily, for 35 days Result:Had antitumor efficacy in a dose-dependent manner.
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    PARP
  • Recptor
    PARP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2589531-76-8
  • Formula Weight
    406.48
  • Molecular Formula
    C22H26N6O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:41.67 mg/mL (102.51 mM; Need ultrasonic)
  • SMILES
    O=C(C1=NC=C(N2CCN(CC3=CC(N4)=C(N=C3)C=C(CC)C4=O)CC2)C=C1)NC
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

molnova catalog
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