AZD5305

CAS No. 2589531-76-8

AZD5305( —— )

Catalog No. M24160 CAS No. 2589531-76-8

AZD5305 is a potent, selective and oral active PARP inhibitor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 258 In Stock
5MG 235 In Stock
10MG 377 In Stock
25MG 630 In Stock
50MG 879 In Stock
100MG 1190 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    AZD5305
  • Note
    Research use only, not for human use.
  • Brief Description
    AZD5305 is a potent, selective and oral active PARP inhibitor.
  • Description
    AZD5305 is a potent, selective and oral active PARP inhibitor.
  • In Vitro
    ——
  • In Vivo
    Animal Model:Female Han Wistar rats with BRCAm xenograft and PDX models (12-13 weeks of age)Dosage:0.01, 0.03, 0.1, and 0.3 mg/kg Administration:Oral administration; daily, for 35 days Result:Had antitumor efficacy in a dose-dependent manner.
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    PARP
  • Recptor
    PARP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2589531-76-8
  • Formula Weight
    406.48
  • Molecular Formula
    C22H26N6O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:41.67 mg/mL (102.51 mM; Need ultrasonic)
  • SMILES
    O=C(C1=NC=C(N2CCN(CC3=CC(N4)=C(N=C3)C=C(CC)C4=O)CC2)C=C1)NC
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

molnova catalog
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