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LY900009
CAS No. 209984-68-9
LY900009( —— )
Catalog No. M23950 CAS No. 209984-68-9
LY900009 is a small molecule inhibitor of Notch signalling via selective inhibition of the γ-secretase protein.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 70 | In Stock |
|
| 5MG | 115 | In Stock |
|
| 10MG | 182 | In Stock |
|
| 25MG | 327 | In Stock |
|
| 50MG | 485 | In Stock |
|
| 100MG | 700 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLY900009
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NoteResearch use only, not for human use.
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Brief DescriptionLY900009 is a small molecule inhibitor of Notch signalling via selective inhibition of the γ-secretase protein.
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DescriptionLY900009 is a small molecule inhibitor of Notch signalling via selective inhibition of the γ-secretase protein.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayNeuroscience
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TargetGamma-secretase
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Recptorγ secretase
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Research Area——
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Indication——
Chemical Information
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CAS Number209984-68-9
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Formula Weight409.49
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Molecular FormulaC23H27N3O4
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Purity>98% (HPLC)
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SolubilityDMSO:10 mM
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SMILESC[C@@H](C(=O)N[C@H]1C2=CC=CC=C2C3=CC=CC=C3N(C1=O)C)NC(=O)[C@H](C(C)C)O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.A first-in-human phase I study of the oral Notch inhibitor, LY900009, in patients with advanced cancer[J]. European Journal of Cancer, 2016, 56.
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