Trifluoperazine

CAS No. 117-89-5

Trifluoperazine( —— )

Catalog No. M21637 CAS No. 117-89-5

Trifluoperazine is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM) and Treatment of schizophrenia.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 46 In Stock
5MG 70 In Stock
10MG 105 In Stock
25MG 192 In Stock
50MG 294 In Stock
100MG 445 In Stock
200MG 641 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Trifluoperazine
  • Note
    Research use only, not for human use.
  • Brief Description
    Trifluoperazine is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM) and Treatment of schizophrenia.
  • Description
    Trifluoperazine is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM) and Treatment of schizophrenia.(In Vitro):Trifluoperazine dihydrochloride is a long-established, widely used 'conventional' antipsychotic agent. Trifluoperazine dihydrochloride has been an extensively studied drug molecule that has been used as a calmodulin inhibitor.Trifluoperazine dihydrochloride acts as a reversible inhibitor of influenza virus morphogenesis, but not budding, by disturbing cellular CaM and/or CaM-dependent functions.
  • In Vitro
    Trifluoperazine is a long-established, widely used 'conventional' antipsychotic agent. Trifluoperazine has been an extensively studied drug molecule that has been used as a calmodulin inhibitor.Trifluoperazine acts as a reversible inhibitor of influenza virus morphogenesis, but not budding, by disturbing cellular CaM and/or CaM-dependent functions.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Dopamine Receptor
  • Recptor
    D2
  • Research Area
    Cardiovascular Disease
  • Indication
    Diamond Blackfan AnemiaPure Red Cell Aplasia

Chemical Information

  • CAS Number
    117-89-5
  • Formula Weight
    407.5
  • Molecular Formula
    C21H24F3N3S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CN1CCN(CCCN2c3ccccc3Sc3ccc(cc23)C(F)(F)F)CC1
  • Chemical Name
    10-[3-(4-methylpiperazin-1-yl)propyl]-2-(trifluoromethyl)phenothiazine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Magdolna Tardy Markuset al. Trifluoperazine versus low-potency first-generation antipsychotic drugs for schizophrenia[J]. Cochrane Database of Systematic Reviews 2014.
molnova catalog
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