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TAPI-1
CAS No. 171235-71-5
TAPI-1( TAPI-1 | TNF-alpha Protease Inhibitor-1 )
Catalog No. M18119 CAS No. 171235-71-5
TAPI-1, an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 25MG | 1476 | In Stock |
|
| 50MG | 2232 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameTAPI-1
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NoteResearch use only, not for human use.
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Brief DescriptionTAPI-1, an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.
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DescriptionTAPI-1 is and inhibitor of TACE. It inhibits the cleavage of TNF-a, TNFRI (p60), and TNFRII (p80).
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In Vitro——
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In Vivo——
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SynonymsTAPI-1 | TNF-alpha Protease Inhibitor-1
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PathwayGPCR/G Protein
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TargetGHSR
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RecptorADAM17/TACE
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number171235-71-5
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Formula Weight499.6
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Molecular FormulaC26H37N5O5
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Purity>98% (HPLC)
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Solubility——
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SMILESCC(C)CC(CC(=O)NO)C(=O)N[C@@H](Cc1cc2ccccc2cc1)C(=O)N[C@@H](C)C(=O)NCCN
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Chemical NameN-[(2S)-1-[[(2S)-1-(2-Aminoethylamino)-1-oxopropan-2-yl]amino]-3-naphthalen-2-yl-1-oxopropan-2-yl]-N'-hydroxy-2-(2-methylpropyl)butanediamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Müllberg J, et al. J Immunol. 1995, 155(11), 5198-5205.
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