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JNJ-63533054

CAS No. 1802326-66-4

JNJ-63533054( JNJ 63533054 | JNJ63533054 | JNJ-63533054 )

Catalog No. M17383 CAS No. 1802326-66-4

JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	65	In Stock
5MG	57	In Stock
10MG	85	In Stock
25MG	170	In Stock
50MG	268	In Stock
100MG	434	In Stock
200MG	622	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

JNJ-63533054
Note

Research use only, not for human use.
Brief Description

JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.
Description

JNJ 63533054 is a potent and selective GPR139 agonist (EC50 = 16 nM) that is brain and cell penetrant. JNJ 63533054 is selective for GPR139 over a panel of GPCRs, ion channels and transporters, including GPR142 and is orally bioavailable.
In Vitro

——
In Vivo

——
Synonyms

JNJ 63533054 | JNJ63533054 | JNJ-63533054
Pathway

Angiogenesis
Target

Adrenergic Receptor
Recptor

hGPR139
Research Area

Neurological Disease
Indication

——

Chemical Information

CAS Number

1802326-66-4
Formula Weight

316.78
Molecular Formula

C17H17ClN2O2
Purity

>98% (HPLC)
Solubility

DMSO : ≥ 50 mg/mL 157.84 mM; H2O : < 0.1 mg/mL
SMILES

C[C@@H](c1ccccc1)NC(=O)CNC(=O)c1cc(ccc1)Cl
Chemical Name

3-Chloro-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Dvorak CA, et al. ACS Med Chem Lett. 2015 Jul 20;6(9):1015-8.

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