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Phentolamine
CAS No. 50-60-2
Phentolamine( —— )
Catalog No. M21648 CAS No. 50-60-2
Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 42 | In Stock |
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| 5MG | 39 | In Stock |
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| 50MG | 110 | In Stock |
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| 100MG | 166 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePhentolamine
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NoteResearch use only, not for human use.
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Brief DescriptionPhentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist.
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DescriptionPhentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist.
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In Vitro——
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In VivoPhentolamine (5-20 mg/kg; i.p.) effectively inhibits the seizures elicited by strychnine (2 mg/kg, i.p.) and attenuates the seizure-potentiating effect of DOPS (4 mg/kg, i.p.) in mouse.Phentolamine (1 mg/kg; i.p.) increases insulin secretion by inhibition of b-cell a2A-adrenoceptors in mouse. Animal Model:WT miceDosage:1 mg/kg Administration:IP Result:Reduced blood glucose and increased insulin levels.
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Synonyms——
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PathwayAngiogenesis
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TargetAdrenergic Receptor
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Recptorα1-adrenergic receptor|α2-adrenergic receptor
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Research AreaOthers
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IndicationDecrease in Night VisionDisturbance
Chemical Information
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CAS Number50-60-2
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Formula Weight281.36
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Molecular FormulaC17H19N3O
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Purity>98% (HPLC)
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Solubility——
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SMILESCc1ccc(cc1)N(CC1=NCCN1)c1cccc(O)c1
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Chemical NamePhenol 3-(((45-dihydro-1H-imidazol-2-yl)methyl)(4-methylphenyl)amino)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Goldstein I. Oral phentolamine: an alpha-1 alpha-2 adrenergic antagonist for the treatment of erectile dysfunction[J]. international journal of impotence research 2000 12:0-0.
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