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DCBS152A
CAS No. ——
DCBS152A( DCBS 152A )
Catalog No. M17022 CAS No. ——
DCBS152A is a potent, functionally selectiver negative modulator of GABAA receptor at the modulatory PQ site in some receptor isoforms.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameDCBS152A
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NoteResearch use only, not for human use.
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Brief DescriptionDCBS152A is a potent, functionally selectiver negative modulator of GABAA receptor at the modulatory PQ site in some receptor isoforms.
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DescriptionDCBS152A is a potent, functionally selectiver negative modulator of GABAA receptor at the modulatory PQ site in some receptor isoforms.
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In Vitro——
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In Vivo——
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SynonymsDCBS 152A
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PathwayMembrane Transporter/Ion Channel
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TargetGAT
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RecptorGAT
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Research Area——
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Indication——
Chemical Information
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CAS Number——
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Formula Weight339.735
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Molecular FormulaC17H10ClN3O3
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name3-(8-chloro-3-oxo-2H,3H,5H-pyrazolo[4,3-c]quinolin-2-yl)benzoic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Treven M, et al. Br J Pharmacol. 2018 Feb;175(3):419-428.
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