Cart
sales@molnova.com
(R)-Baclofen
CAS No. 69308-37-8
(R)-Baclofen( STX-209 )
Catalog No. M15651 CAS No. 69308-37-8
A derivative of the neurotransmitter GABA that acts as a GABAB receptor agonist; also blocks α2δ subunit-containing voltage-dependent calcium channel (VDCC) with Ki of 156 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 30 | In Stock |
|
| 10MG | 50 | In Stock |
|
| 25MG | 106 | In Stock |
|
| 50MG | 176 | In Stock |
|
| 100MG | 272 | In Stock |
|
| 200MG | 388 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product Name(R)-Baclofen
-
NoteResearch use only, not for human use.
-
Brief DescriptionA derivative of the neurotransmitter GABA that acts as a GABAB receptor agonist; also blocks α2δ subunit-containing voltage-dependent calcium channel (VDCC) with Ki of 156 uM.
-
DescriptionA derivative of the neurotransmitter GABA that acts as a GABAB receptor agonist; also blocks α2δ subunit-containing voltage-dependent calcium channel (VDCC) with Ki of 156 uM; A neurotransmitter inhibitor by blocking the release of excitatory transmitters; serves as a central nervous system depressant and skeletal muscle relaxant.Other Indication Approved.
-
In Vitro——
-
In Vivo——
-
SynonymsSTX-209
-
PathwayMembrane Transporter/Ion Channel
-
TargetGAT
-
RecptorGABAR
-
Research AreaOther Indications
-
IndicationOther Disease
Chemical Information
-
CAS Number69308-37-8
-
Formula Weight213.6608
-
Molecular FormulaC10H12ClNO2
-
Purity>98% (HPLC)
-
SolubilityH2O: 5 mg/mL (Need ultrasonic)
-
SMILESO=C(O)C[C@H](C1=CC=C(Cl)C=C1)CN
-
Chemical NameBenzenepropanoic acid, β-(aminomethyl)-4-chloro-, (βR)-
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Zvejniece L, et al. Pharmacol Biochem Behav. 2015 Oct;137:23-9.
2. Carter LP, et al. Pharmacol Ther. 2009 Jan;121(1):100-14.
molnova catalog
related products
-
Alprazolam
Alprazolam (D-65MT;U 31889) is a triazolobenzodiazepine agent with anxiolytic, sedative-hypnotic and anticonvulsant activities.
-
Pentetrazol
Pentylenetetrazol is a GABA(A) receptor antagonist, kindles model of epilepsy.
-
Tiagabine
Tiagabine hydrochloride(NO328 hydrochloride) is a selective gamma-aminobutyric acid (GABA) reuptake inhibitor.
