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Home - Products - GPCR/G Protein - Cannabinoid Receptor - A 834735

A 834735

CAS No. 895155-57-4

A 834735( A-834735 | A834735 )

Catalog No. M16446 CAS No. 895155-57-4

A potent, nonselective, brain penetrant, full agonist at both the central CB1 and peripheral CB2 receptors with Ki of 4.6 and 0.31 nM, respectively.

Purity : >98% (HPLC)

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Biological Information

  • Product Name
    A 834735
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, nonselective, brain penetrant, full agonist at both the central CB1 and peripheral CB2 receptors with Ki of 4.6 and 0.31 nM, respectively.
  • Description
    A potent, nonselective, brain penetrant, full agonist at both the central CB1 and peripheral CB2 receptors with Ki of 4.6 and 0.31 nM, respectively; reverses thermal hyperalgesia without adverse side effects in a rat neuropathic pain model.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    A-834735 | A834735
  • Pathway
    GPCR/G Protein
  • Target
    Cannabinoid Receptor
  • Recptor
    Cannabinoid Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    895155-57-4
  • Formula Weight
    339.5
  • Molecular Formula
    C22H29NO2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C(C1=CN(CC2CCOCC2)C3=C1C=CC=C3)C4C(C)(C)C4(C)C
  • Chemical Name
    [1-[(tetrahydro-2H-pyran-4-yl)methyl]-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)-methanone

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Chin CL, et al. Br J Pharmacol. 2008 Jan;153(2):367-79. 2. Grim TW, et al. J Pharmacol Exp Ther. 2016 Nov;359(2):329-339.
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