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A 834735
CAS No. 895155-57-4
A 834735( A-834735 | A834735 )
Catalog No. M16446 CAS No. 895155-57-4
A potent, nonselective, brain penetrant, full agonist at both the central CB1 and peripheral CB2 receptors with Ki of 4.6 and 0.31 nM, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameA 834735
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, nonselective, brain penetrant, full agonist at both the central CB1 and peripheral CB2 receptors with Ki of 4.6 and 0.31 nM, respectively.
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DescriptionA potent, nonselective, brain penetrant, full agonist at both the central CB1 and peripheral CB2 receptors with Ki of 4.6 and 0.31 nM, respectively; reverses thermal hyperalgesia without adverse side effects in a rat neuropathic pain model.
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In Vitro——
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In Vivo——
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SynonymsA-834735 | A834735
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PathwayGPCR/G Protein
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TargetCannabinoid Receptor
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RecptorCannabinoid Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number895155-57-4
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Formula Weight339.5
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Molecular FormulaC22H29NO2
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(C1=CN(CC2CCOCC2)C3=C1C=CC=C3)C4C(C)(C)C4(C)C
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Chemical Name[1-[(tetrahydro-2H-pyran-4-yl)methyl]-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)-methanone
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Chin CL, et al. Br J Pharmacol. 2008 Jan;153(2):367-79.
2. Grim TW, et al. J Pharmacol Exp Ther. 2016 Nov;359(2):329-339.
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