IKK-16 (IKK Inhibitor VII)

CAS No. 873225-46-8

IKK-16 (IKK Inhibitor VII)( —— )

Catalog No. M16348 CAS No. 873225-46-8

IKK-16 (IKK Inhibitor VII) is a selective IκB kinase (IKK) inhibitor for IKK-2, IKK complex and IKK-1 with IC50 of 40 nM, 70 nM and 200 nM, respectively.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 85 In Stock
2MG 46 In Stock
5MG 76 In Stock
10MG 135 In Stock
25MG 245 In Stock
50MG 398 In Stock
100MG 569 In Stock
200MG 807 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    IKK-16 (IKK Inhibitor VII)
  • Note
    Research use only, not for human use.
  • Brief Description
    IKK-16 (IKK Inhibitor VII) is a selective IκB kinase (IKK) inhibitor for IKK-2, IKK complex and IKK-1 with IC50 of 40 nM, 70 nM and 200 nM, respectively.
  • Description
    IKK-16 (IKK Inhibitor VII) is a selective IκB kinase (IKK) inhibitor for IKK-2, IKK complex and IKK-1 with IC50 of 40 nM, 70 nM and 200 nM, respectively.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Immunology/Inflammation
  • Target
    IκB kinase (IKK)
  • Recptor
    IKK2| IKK1| IKK complex
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    873225-46-8
  • Formula Weight
    483.63
  • Molecular Formula
    C??H??N?OS
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:90 mg/mL (186.1 mM);Ethanol:<1 mg/mL;Water:<1 mg/mL
  • SMILES
    O=C(N1CCC(CC1)N1CCCC1)C1=CC=C(NC2=NC=CC(=N2)C2=CC3=CC=CC=C3S2)C=C1 |c:22,24,31,33,38,t:15,17,20,27,29|
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Waelchli R, et al. Bioorg Med Chem Lett, 2006, 16(1), 108-112.
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