Azilsartan medoxomil monopotassium

CAS No. 863031-24-7

Azilsartan medoxomil monopotassium( TAK-491 )

Catalog No. M16247 CAS No. 863031-24-7

An orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 32 In Stock
5MG 54 In Stock
10MG 82 In Stock
25MG 164 In Stock
50MG 242 In Stock
100MG 356 In Stock
200MG 507 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Azilsartan medoxomil monopotassium
  • Note
    Research use only, not for human use.
  • Brief Description
    An orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM.
  • Description
    An orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. Hypertension Approved.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    TAK-491
  • Pathway
    GPCR/G Protein
  • Target
    Angiotensin Receptor
  • Recptor
    Angiotensin Receptor
  • Research Area
    Cardiovascular Disease
  • Indication
    Hypertension

Chemical Information

  • CAS Number
    863031-24-7
  • Formula Weight
    606.6239
  • Molecular Formula
    C30H23KN4O8
  • Purity
    >98% (HPLC)
  • Solubility
    10 mM in DMSO
  • SMILES
    CCOC1=NC2=CC=CC(=C2N1CC3=CC=C(C=C3)C4=CC=CC=C4C5=NC(=O)O[N-]5)C(=O)OCC6=C(OC(=O)O6)C.[K+]
  • Chemical Name
    1H-Benzimidazole-7-carboxylic acid, 1-[[2'-(2,5-dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-, (5-methyl-2-oxo-1,3-dioxol-4-yl)methyl ester, potassium salt (1:1)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

molnova catalog
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