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Nefopam hydrochloride
CAS No. 23327-57-3
Nefopam hydrochloride( —— )
Catalog No. M13669 CAS No. 23327-57-3
Nefopam hydrochloride is a centrally-acting but non-opioid analgesic drug by blocking voltage-gated sodium channel and inhibition of serotonin, dopamine and noradrenaline reuptake.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 34 | In Stock |
|
| 1G | 54 | In Stock |
|
Biological Information
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Product NameNefopam hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionNefopam hydrochloride is a centrally-acting but non-opioid analgesic drug by blocking voltage-gated sodium channel and inhibition of serotonin, dopamine and noradrenaline reuptake.
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DescriptionNefopam hydrochloride is a centrally-acting but non-opioid analgesic drug by blocking voltage-gated sodium channel and inhibition of serotonin, dopamine and noradrenaline reuptake.(In Vitro):Nefopam hydrochloride (Fenazoxine hydrochloride) is a non-opioid, non-steroidal, centrally acting analgesic drug that is derivative of the non-sedative benzoxazocine. Constitutively elevated β-catenin leads to a delayed and fibrous fracture repair process, and Nefopam inhibits β-catenin mediated signaling during skin wound repair.
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In VitroNefopam hydrochloride (Fenazoxine hydrochloride) is a non-opioid, non-steroidal, centrally acting analgesic drug that is derivative of the non-sedative benzoxazocine.Constitutively elevated β-catenin leads to a delayed and fibrous fracture repair process, and Nefopam inhibits β-catenin mediated signaling during skin wound repair.
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In Vivo——
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetSodium Channel
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RecptorSodium Channel
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Research AreaNeurological Disease
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Indication——
Chemical Information
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CAS Number23327-57-3
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Formula Weight289.8
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Molecular FormulaC17H20ClNO
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Purity>98% (HPLC)
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SolubilityWater: 21 mg/mL (72.46 mM); DMSO: 1 mg/mL (3.45 mM)
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SMILESCl.CN1CCOC(C2=CC=CC=C2)C2=CC=CC=C2C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. M. S. Evans1, et al, lBr J Anaesth, 2008, 101(5), 610-617.
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