Cart
sales@molnova.com
MS012
CAS No. 2089617-83-2
MS012( MS 012 )
Catalog No. M13271 CAS No. 2089617-83-2
MS012 is a potent and selective inhibitor of G9a-Like Protein (GLP) lysine methyltransferase with IC50 of 7 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameMS012
-
NoteResearch use only, not for human use.
-
Brief DescriptionMS012 is a potent and selective inhibitor of G9a-Like Protein (GLP) lysine methyltransferase with IC50 of 7 nM.
-
DescriptionMS012 is a potent and selective inhibitor of G9a-Like Protein (GLP) lysine methyltransferase with IC50 of 7 nM, shows >30-fold selectivity for GLP over G9a and other methyltransferases.
-
In Vitro——
-
In Vivo——
-
SynonymsMS 012
-
PathwayChromatin/Epigenetic
-
TargetHMTase
-
RecptorHMTase
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number2089617-83-2
-
Formula Weight401.555
-
Molecular FormulaC22H35N5O2
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESCOC1=CC2=NC(NCCCCCC)=NC(NC3CCN(C)CC3)=C2C=C1OC
-
Chemical NameN2-Hexyl-6,7-dimethoxy-N4-(1-methylpiperidin-4-yl)quinazoline2,4-diamine
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Xiong Y, et al. J Med Chem. 2017 Mar 9;60(5):1876-1891.
molnova catalog
related products
-
JQEZ-5
A novel potent, selective, SAM-competitive EZH2 inhibitor with IC50 of 80 nM (inhibition of enzymatic function of PRC2).
-
3-Deazaneplanocin A
A highly potent and competitive S-adenosylhomocysteine hydrolase inhibitor with Ki of 0.05 nM.
-
PFI-2
A first-in-class, potent and selective inhibitor of SETD7 methyltransferase with Ki app/IC50 of 0.33/2 nM.
