BETi-211( BETi 211 | BETi211 )

Catalog No. M13114 CAS No. 1995867-02-1

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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Product Name

BETi-211
Note

Research use only, not for human use.
Brief Description

A novel potent small-molecule BET bromodomain (BRD) inhibitor that binds to BET proteins with Ki values of <1 nM.
Description

A novel potent small-molecule BET bromodomain (BRD) inhibitor that binds to BET proteins with Ki values of <1 nM; exhibits >10-100 times more potent than RX-37, JQ-1, OTX-015 or IBET-762.
In Vitro

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In Vivo

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Synonyms

BETi 211 | BETi211
Pathway

Chromatin/Epigenetic
Target

Bromodomain
Recptor

Bromodomain
Research Area

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Indication

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CAS Number

1995867-02-1
Formula Weight

487.564
Molecular Formula

C26H29N7O3
Purity

>98% (HPLC)
Solubility

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SMILES

COCC1=NC(NC2=CC(C3CC3)=NN2CC)=C4C(NC5=C4C=C(OC)C(C6=C(C)ON=C6C)=C5)=N1
Chemical Name

N-(3-cyclopropyl-1-ethyl-1H-pyrazol-5-yl)-7-(3,5-dimethylisoxazol-4-yl)-6-methoxy-2-(methoxymethyl)-9H-pyrimido[4,5-b]indol-4-amine