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Atazanavir
CAS No. 198904-31-3
Atazanavir( BMS-232632 )
Catalog No. M13109 CAS No. 198904-31-3
A highly potent HIV-1 protease inhibitor that exhibits potent anti-HIV activity EC50 of 2.6-5.3 nM and EC90 of 9-15 nM in cell culture.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 35 | In Stock |
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| 10MG | 57 | In Stock |
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| 25MG | 86 | In Stock |
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| 50MG | 113 | In Stock |
|
| 100MG | 194 | In Stock |
|
| 200MG | 291 | In Stock |
|
| 500MG | 492 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameAtazanavir
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NoteResearch use only, not for human use.
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Brief DescriptionA highly potent HIV-1 protease inhibitor that exhibits potent anti-HIV activity EC50 of 2.6-5.3 nM and EC90 of 9-15 nM in cell culture.
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DescriptionA highly potent HIV-1 protease inhibitor that exhibits potent anti-HIV activity EC50 of 2.6-5.3 nM and EC90 of 9-15 nM in cell culture; shows synergistic antiviral effects in HIV-infected PBMCs; used to treat and prevent HIV/AIDS.HIV Infection Approved.
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In Vitro——
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In Vivo——
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SynonymsBMS-232632
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PathwayMicrobiology/Virology
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TargetHIV
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RecptorHIVProtease
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Research AreaInfection
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IndicationHIV Infection
Chemical Information
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CAS Number198904-31-3
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Formula Weight704.8555
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Molecular FormulaC38H52N6O7
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESCC(C)(C)[C@@H](C(=O)N[C@@H](CC1=CC=CC=C1)[C@H](CN(CC2=CC=C(C=C2)C3=CC=CC=N3)NC(=O)[C@H](C(C)(C)C)NC(=O)OC)O)NC(=O)OC
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Chemical Name2,5,6,10,13-Pentaazatetradecanedioic acid, 3,12-bis(1,1-dimethylethyl)-8-hydroxy-4,11-dioxo-9-(phenylmethyl)-6-[[4-(2-pyridinyl)phenyl]methyl]-, 1,14-dimethyl ester, (3S,8S,9S,12S)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Robinson BS, et al. Antimicrob Agents Chemother. 2000 Aug;44(8):2093-9.
2. Gong YF, et al. Antimicrob Agents Chemother. 2000 Sep;44(9):2319-26.
3. Drusano GL, et al. J Infect Dis. 2001 Apr 1;183(7):1126-9.
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