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Semaxanib
CAS No. 194413-58-6
Semaxanib ( SU5416 )
Catalog No. M13045 CAS No. 194413-58-6
Semaxanib (SU5416) is a potent and selective VEGFR(Flk-1/KDR) inhibitor with IC50 of 1.23 μM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 37 | In Stock |
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| 10MG | 30 | In Stock |
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| 25MG | 48 | In Stock |
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| 50MG | 71 | In Stock |
|
| 100MG | 111 | In Stock |
|
| 200MG | 174 | In Stock |
|
| 500MG | 341 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSemaxanib
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NoteResearch use only, not for human use.
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Brief DescriptionSemaxanib (SU5416) is a potent and selective VEGFR(Flk-1/KDR) inhibitor with IC50 of 1.23 μM.
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DescriptionSemaxanib (SU5416) is a potent and selective VEGFR(Flk-1/KDR) inhibitor with IC50 of 1.23 μM, 20-fold more selective for VEGFR than PDGFRβ, lack of activity against EGFR, InsR and FGFR. Phase 3.
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In Vitro——
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In Vivo——
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SynonymsSU5416
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PathwayAngiogenesis
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TargetVEGFR
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RecptorVEGFR2/Flk1
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number194413-58-6
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Formula Weight238.28
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Molecular FormulaC15H14N2O
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Purity>98% (HPLC)
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SolubilityEthanol: 2 mg/mL (8.39 mM); DMSO: 22 mg/mL (92.32 mM)
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SMILESCC1=CC(=C(N1)/C=C\2/C3=CC=CC=C3NC2=O)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Fong TA, et al. Y Res, 1999, 59(1), 99-106.
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