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MAP4K4-IN-17
CAS No. 1811510-58-3
MAP4K4-IN-17( —— )
Catalog No. M12780 CAS No. 1811510-58-3
MAP4K4-IN-17 is a potent and highly selective MAP4K4 inhibitor with IC50 of 14.9 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 41 | In Stock |
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| 5MG | 37 | In Stock |
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| 10MG | 68 | In Stock |
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| 25MG | 147 | In Stock |
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| 50MG | 230 | In Stock |
|
| 100MG | 365 | In Stock |
|
| 200MG | 541 | In Stock |
|
| 500MG | 823 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameMAP4K4-IN-17
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NoteResearch use only, not for human use.
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Brief DescriptionMAP4K4-IN-17 is a potent and highly selective MAP4K4 inhibitor with IC50 of 14.9 nM.
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DescriptionMAP4K4-IN-17 is a potent and highly selective MAP4K4 inhibitor with IC50 of 14.9 nM, showes improved overall drug-like properties compared to PF-06260933; a lead compound for advanced preclinical development.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMAPK/ERK Signaling
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TargetMAP4K
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RecptorMAP4K
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Research Area——
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Indication——
Chemical Information
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CAS Number1811510-58-3
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Formula Weight297.746
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Molecular FormulaC15H12ClN5
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 10 mg/mL (33.59 mM)
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SMILES——
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Chemical Name5-(6-amino-5-(4-chlorophenyl)pyridin-3-yl)pyrimidin-2-amine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ammirati M, et al. ACS Med Chem Lett. 2015 Oct 6;6(11):1128-33.
molnova catalog
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