PU-H54

CAS No. 1454619-13-6

PU-H54( PU H 54 )

Catalog No. M11959 CAS No. 1454619-13-6

A potent, selective Grp94 inhibitor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 69 In Stock
10MG 112 In Stock
25MG 259 In Stock
50MG 375 In Stock
100MG 533 In Stock
200MG 724 In Stock
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Biological Information

  • Product Name
    PU-H54
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, selective Grp94 inhibitor.
  • Description
    A potent, selective Grp94 inhibitor.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    PU H 54
  • Pathway
    Cytoskeleton/Cell Adhesion Molecules
  • Target
    HSP
  • Recptor
    HSP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1454619-13-6
  • Formula Weight
    337.45
  • Molecular Formula
    C18H19N5S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (296.35 mM)
  • SMILES
    CC1=CC(C)=C(SC2=NC3=C(N)N=CN(CCCC#C)C3=N2)C=C1
  • Chemical Name
    8-((2,4-dimethylphenyl)thio)-3-(pent-4-yn-1-yl)-3H-purin-6-amine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Khandelwal A, et al. ACS Med Chem Lett. 2017 Sep 1;8(10):1013-1018. 2. Crowley VM, et al. J Med Chem. 2016 Apr 14;59(7):3471-88.
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