Cart
sales@molnova.com
XL-001
CAS No. 1426153-46-9
XL-001( XL001 )
Catalog No. M11799 CAS No. 1426153-46-9
XL-001 (XL001) is a novel specific CB2 inverse agonist with Ki of 0.5 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameXL-001
-
NoteResearch use only, not for human use.
-
Brief DescriptionXL-001 (XL001) is a novel specific CB2 inverse agonist with Ki of 0.5 nM.
-
DescriptionXL-001 (XL001) is a novel specific CB2 inverse agonist with Ki of 0.5 nM; inhibits in a dose-dependent fashion the fibrogenic response induced by CB2 overexpression, CB2 agonist or transforming growth factor-β1, ameliorates kidney injury, fibrosis and inflammation in both the obstruction and ischemia/reperfusion models.
-
In Vitro——
-
In Vivo——
-
SynonymsXL001
-
PathwayGPCR/G Protein
-
TargetCannabinoid Receptor
-
RecptorCannabinoid Receptor
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number1426153-46-9
-
Formula Weight438.586
-
Molecular FormulaC25H30N2O3S
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESCCN(CC)C1=CC=C(C=C1)CN(C2=CC=C(C=C2)C)S(=O)(=O)C3=CC=C(C=C3)OC
-
Chemical NameN-(4-(diethylamino)benzyl)-4-methoxy-N-(p-tolyl)benzenesulfonamide
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Zhou L, et al. Kidney Int. 2018 Aug 6. pii: S0085-2538(18)30397-1.
molnova catalog
related products
-
VCE-004.3
VCE-004.3 (VCE004.3) is a novel semi-synthetic cannabidiol derivative behaving as a dual PPARγ/CB2 agonist and CB1 receptor modulator.
-
NESS-0327
A potent, selective CB1 cannabinoid receptor antagonist with Ki of 350 fM.
-
CB1 inverse agonist ...
CB1 inverse agonist 1 (MRL-650) is an orally active and selective CB1 agonist. The IC50s for CB1 and CB2 are 7.5 nM and 4100 nM, respectively.
