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BMS 830216

CAS No. 1197420-06-6

BMS 830216( BMS-830216 | BMS830216 )

Catalog No. M10704 CAS No. 1197420-06-6

The the phosphate ester prodrug of BMS 819881, a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    BMS 830216
  • Note
    Research use only, not for human use.
  • Brief Description
    The the phosphate ester prodrug of BMS 819881, a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.
  • Description
    The the phosphate ester prodrug of BMS 819881, a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM; shows potential for treatment of obesity.ObesityPhase 2 Discontinued.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    BMS-830216 | BMS830216
  • Pathway
    GPCR/G Protein
  • Target
    MCHR
  • Recptor
    MCHR
  • Research Area
    Metabolic Disease
  • Indication
    Obesity

Chemical Information

  • CAS Number
    1197420-06-6
  • Formula Weight
    548.931
  • Molecular Formula
    C24H22ClN2O7PS
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    COC1=C(C=CC(=C1)N2C=NC3=C(C2=O)SC(=C3)C4=CC=C(C=C4)Cl)OCC(C5CC5)OP(=O)(O)O
  • Chemical Name
    (R)-2-(4-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-2-methoxyphenoxy)-1-cyclopropylethyl dihydrogen phosphate

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Washburn WN, et al. J Med Chem. 2014 Sep 25;57(18):7509-22.
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