Cart
sales@molnova.com
PK-14105
CAS No. 107257-28-3
PK-14105( PK14105 )
Catalog No. M10296 CAS No. 107257-28-3
A potent photoaffinity ligand for the peripheral-type benzodiazepine binding site with Ki of 4 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 195 | Get Quote |
|
| 50MG | 851 | Get Quote |
|
| 100MG | 1341 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NamePK-14105
-
NoteResearch use only, not for human use.
-
Brief DescriptionA potent photoaffinity ligand for the peripheral-type benzodiazepine binding site with Ki of 4 nM.
-
DescriptionA potent photoaffinity ligand for the peripheral-type benzodiazepine binding site with Ki of 4 nM; attaches covalently and specifically to all the PBS when cardiac membranes are irradiated with this compound under ultraviolet light.
-
In Vitro——
-
In Vivo——
-
SynonymsPK14105
-
PathwayMembrane Transporter/Ion Channel
-
TargetGAT
-
RecptorGAT
-
Research AreaOther Indications
-
Indication——
Chemical Information
-
CAS Number107257-28-3
-
Formula Weight381.4002
-
Molecular FormulaC21H20FN3O3
-
Purity>98% (HPLC)
-
SolubilityDMSO: ≥ 30 mg/mL
-
SMILESO=C(C1=CC2=C(C(C3=CC([N+]([O-])=O)=CC=C3F)=N1)C=CC=C2)N(C(CC)C)C
-
Chemical Name3-Isoquinolinecarboxamide, 1-(2-fluoro-5-nitrophenyl)-N-methyl-N-(1-methylpropyl)-
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Doble A, et al. Mol Pharmacol. 1987 Jan;31(1):42-9.
2. Doble A, et al. J Recept Res. 1987;7(1-4):55-70.
3. Skowroński R, et al. Eur J Pharmacol. 1988 Mar 29;148(2):187-93.
molnova catalog
related products
-
AZD6280
AZD6280 is a potent, α2/3 functionally selective, partial GABAA receptor modulator with pKi of 7.7.
-
DCBS152A
DCBS152A is a potent, functionally selectiver negative modulator of GABAA receptor at the modulatory PQ site in some receptor isoforms.
-
4-Aminobutyric acid
The most common inhibitory neurotransmitter in the central nervous system.
