Cart
sales@molnova.com
LY2183240
CAS No. 874902-19-9
LY2183240 ( —— )
Catalog No. M24889 CAS No. 874902-19-9
LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 270 pM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 35 | In Stock |
|
| 10MG | 58 | In Stock |
|
| 25MG | 120 | In Stock |
|
| 50MG | 228 | In Stock |
|
| 100MG | 356 | In Stock |
|
| 500MG | 836 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameLY2183240
-
NoteResearch use only, not for human use.
-
Brief DescriptionLY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 270 pM).
-
DescriptionLY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 270 pM).
-
Synonyms——
-
PathwayAutophagy
-
TargetAutophagy
-
RecptorAutophagy;FAAH
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number874902-19-9
-
Formula Weight307.4
-
Molecular FormulaC17H17N5O
-
Purity>98% (HPLC)
-
SolubilityDMSO:50 mg/mL (162.68 mM; Need ultrasonic)
-
SMILESO=C(N(C)C)N1N=NN=C1CC(C=C2)=CC=C2C3=CC=CC=C3
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Dickason-Chesterfield AK, et al. Pharmacological characterization of endocannabinoid transport and fatty acid amide hydrolase inhibitors. Cell Mol Neurobiol. 2006 Jul-Aug;26(4-6):407-23.
molnova catalog
related products
-
Sulfuretin
Sulfuretin is a potent anti-oxidant, has protective effect against t-BHP-induced oxidative damage in human liver-derived HepG2 cells is attributable to its ability to scavenge ROS and up-regulate the activity of HO-1 through the Nrf2/ARE and JNK/ERK signaling pathways.
-
SLLN-15
SLLN-15 (Autophagy inducer SLLN-15) is a potent, orally available inducer of autophagy that selectively activated cytostatic macroautophagy/autophagy in TNBC preclinical models.
-
Hemin
Hemin, a physiological erythroid maturation stimulator, is able to induce the expression of critical autophagic genes (Map1a1b (LC3), Beclin-1 gen, Atg5) in an erythroleukemia cell type.
