LDN-192960

CAS No. 184582-62-5

LDN-192960 ( —— )

Catalog No. M23838 CAS No. 184582-62-5

LDN-192960 is a potent inhibitor of Haspin and DYRK2 (IC50s: 10 nM and 48 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 147 In Stock
10MG 237 In Stock
25MG 475 In Stock
50MG 692 In Stock
100MG 972 In Stock
500MG 1944 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    LDN-192960
  • Note
    Research use only, not for human use.
  • Brief Description
    LDN-192960 is a potent inhibitor of Haspin and DYRK2 (IC50s: 10 nM and 48 nM).
  • Description
    LDN-192960 is a potent inhibitor of Haspin and DYRK2 (IC50s: 10 nM and 48 nM).
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    DYRK2; Haspin
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    184582-62-5
  • Formula Weight
    328.4
  • Molecular Formula
    C18H20N2O2S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:30 mg/mL (91.34 mM);Water:10 mg/mL (30.45 mM)
  • SMILES
    NCCCSC1=C(C=C(OC)C=C2)C2=NC3=CC=C(OC)C=C31
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Cuny GD, et al. Structure-activity relationship study of acridine analogs as haspin and DYRK2 kinase inhibitors. Bioorg Med Chem Lett. 2010 Jun 15;20(12):3491-4.
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