Ketanserin

CAS No. 74050-98-9

Ketanserin ( R41468 )

Catalog No. M15827 CAS No. 74050-98-9

A high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
25MG 27 In Stock
100MG 43 In Stock
200MG 79 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Ketanserin
  • Note
    Research use only, not for human use.
  • Brief Description
    A high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C.
  • Description
    A high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C; also has a high affinity antagonist for the H1 receptor (Ki= 2 nM) and α1-adrenergic receptor (Ki=40 nM); an antihypertensive agent.Hypertension Approved
  • Synonyms
    R41468
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT2A;5-HT2C(Human);5-HT2C(Rat)
  • Research Area
    Cardiovascular Disease
  • Indication
    Hypertension

Chemical Information

  • CAS Number
    74050-98-9
  • Formula Weight
    395.43
  • Molecular Formula
    C22H22FN3O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 8 mg/mL
  • SMILES
    O=C(N1CCN2CCC(C(C3=CC=C(F)C=C3)=O)CC2)NC4=C(C=CC=C4)C1=O
  • Chemical Name
    2,4(1H,3H)-Quinazolinedione, 3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Creed-Carson M, et al. Behav Brain Res. 2011 Jun 1;219(2):273-9.
2. Catafau AM, et al. J Cereb Blood Flow Metab. 2010 May;30(5):985-93.
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