Ketanserin
CAS No. 74050-98-9
Ketanserin ( R41468 )
Catalog No. M15827 CAS No. 74050-98-9
A high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
25MG | 27 | In Stock |
|
100MG | 43 | In Stock |
|
200MG | 79 | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
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Product NameKetanserin
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NoteResearch use only, not for human use.
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Brief DescriptionA high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C.
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DescriptionA high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C; also has a high affinity antagonist for the H1 receptor (Ki= 2 nM) and α1-adrenergic receptor (Ki=40 nM); an antihypertensive agent.Hypertension Approved
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SynonymsR41468
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT2A;5-HT2C(Human);5-HT2C(Rat)
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Research AreaCardiovascular Disease
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IndicationHypertension
Chemical Information
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CAS Number74050-98-9
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Formula Weight395.43
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Molecular FormulaC22H22FN3O3
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Purity>98% (HPLC)
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SolubilityDMSO: 8 mg/mL
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SMILESO=C(N1CCN2CCC(C(C3=CC=C(F)C=C3)=O)CC2)NC4=C(C=CC=C4)C1=O
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Chemical Name2,4(1H,3H)-Quinazolinedione, 3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Creed-Carson M, et al. Behav Brain Res. 2011 Jun 1;219(2):273-9.
2. Catafau AM, et al. J Cereb Blood Flow Metab. 2010 May;30(5):985-93.
2. Catafau AM, et al. J Cereb Blood Flow Metab. 2010 May;30(5):985-93.
molnova catalog
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