MIN-117
CAS No. 310392-93-9
MIN-117 ( WF-516;WF 516;MIN 117 )
Catalog No. M13993 CAS No. 310392-93-9
A small molecule 5-HT1A and 5-HT2A receptor antagonist and inhibitor of serotonin and dopamine reuptake, also possess affinity for the α1A- and α1B-adrenergic receptors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 1053 | Get Quote |
|
50MG | 2142 | Get Quote |
|
100MG | 2790 | Get Quote |
|
200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
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Product NameMIN-117
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NoteResearch use only, not for human use.
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Brief DescriptionA small molecule 5-HT1A and 5-HT2A receptor antagonist and inhibitor of serotonin and dopamine reuptake, also possess affinity for the α1A- and α1B-adrenergic receptors.
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DescriptionA small molecule 5-HT1A and 5-HT2A receptor antagonist and inhibitor of serotonin and dopamine reuptake, also possess affinity for the α1A- and α1B-adrenergic receptors.Depression Phase 2 Clinical
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SynonymsWF-516;WF 516;MIN 117
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT Receptor
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Research AreaNeurological Disease
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IndicationDepression
Chemical Information
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CAS Number310392-93-9
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Formula Weight538.85
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Molecular FormulaC25H26Cl3N3O4
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Purity>98% (HPLC)
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Solubility——
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SMILESCC1=NN=C(O1)C2=CC3=C(O2)C=CC=C3OCC(CN4CCC(CC4)C5=CC(=C(C=C5)Cl)Cl)O.Cl
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Chemical Name(2S)-1-[4-(3,4-dichlorophenyl)piperidin-1-yl]-3-[2-(5-methyl-1,3,4-oxadiazol-2-yl)benzo[b]furan-4-yloxy]propan-2-ol monohydrochloride
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. El Mansari M, et al. Naunyn Schmiedebergs Arch Pharmacol. 2008 Jan;376(5):351-61.
2. Saijo T, et al. PLoS One. 2012;7(8):e42589. doi: 10.1371/journal.pone.0042589.
2. Saijo T, et al. PLoS One. 2012;7(8):e42589. doi: 10.1371/journal.pone.0042589.
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