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KS-176
CAS No. 1253452-78-6
KS-176( KS 176 | KS176 )
Catalog No. M11019 CAS No. 1253452-78-6
A potent and selective inhibitor of BCRP multidrug transporter with IC50 of 0.59 and 1.39 uM in Pheo A and Hoechst 33342 assays, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 45 | In Stock |
|
| 5MG | 71 | In Stock |
|
| 10MG | 120 | In Stock |
|
| 25MG | 264 | In Stock |
|
| 50MG | 482 | In Stock |
|
| 100MG | 696 | In Stock |
|
| 500MG | 1431 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameKS-176
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NoteResearch use only, not for human use.
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Brief DescriptionA potent and selective inhibitor of BCRP multidrug transporter with IC50 of 0.59 and 1.39 uM in Pheo A and Hoechst 33342 assays, respectively.
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DescriptionA potent and selective inhibitor of BCRP multidrug transporter with IC50 of 0.59 and 1.39 uM in Pheo A and Hoechst 33342 assays, respectively; displays no inhibitory activity against P-gp or MRP1.
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In Vitro——
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In Vivo——
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SynonymsKS 176 | KS176
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PathwayMembrane Transporter/Ion Channel
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TargetBCRP
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RecptorBKCa-channel
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1253452-78-6
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Formula Weight405.4034
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Molecular FormulaC22H19N3O5
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 35 mg/mL
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SMILESO=C(NC1=CC=C(CCO)C=C1)C2=CC=CC=C2NC(C3=CC=C([N+]([O-])=O)C=C3)=O
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Chemical NameBenzamide, N-[4-(2-hydroxyethyl)phenyl]-2-[(4-nitrobenzoyl)amino]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Pick A, et al. ChemMedChem. 2010 Sep 3;5(9):1498-505.
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