KDM4D-IN-10r

CAS No. 2098902-68-0

KDM4D-IN-10r ( —— )

Catalog No. M13322 CAS No. 2098902-68-0

KDM4D-IN-10r is a potent, selective histone lysine demethylase 4D (KDM4D) inhibitor with IC50 of 0.41 uM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 222 In Stock
10MG 361 In Stock
25MG 601 In Stock
50MG 858 In Stock
100MG 1161 In Stock
500MG 2331 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    KDM4D-IN-10r
  • Note
    Research use only, not for human use.
  • Brief Description
    KDM4D-IN-10r is a potent, selective histone lysine demethylase 4D (KDM4D) inhibitor with IC50 of 0.41 uM.
  • Description
    KDM4D-IN-10r is a potent, selective histone lysine demethylase 4D (KDM4D) inhibitor with IC50 of 0.41 uM; has no significant activity against KDM2B, KDM3B, KDM2B (IC50>10 uM).
  • Synonyms
    ——
  • Pathway
    Chromatin/Epigenetic
  • Target
    Histone Demethylase
  • Recptor
    KDM4D
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2098902-68-0
  • Formula Weight
    225.21
  • Molecular Formula
    C11H7N5O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 6 mg/mL, Need Ultrasonic ( < 1 mg/ml refers to the product slightly soluble or insoluble )
  • SMILES
    CC1=NN2C(=C1C#N)NC(=O)C3=C2N=CC=C3
  • Chemical Name
    5-hydroxy-2-methylpyrazolo[1,5-a]pyrido[3,2-e]pyrimidine-3-carbonitrile

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Fang Z, et al. Bioorg Med Chem Lett. 2017 Jul 15;27(14):3201-3204.
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