IDH1-IN-1 ( Mutant IDH1-IN-1 )

Catalog No. M11452 CAS No. 1355326-21-4

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Product Name

IDH1-IN-1
Note

Research use only, not for human use.
Brief Description

Mutant IDH1-IN-1 is a potent mutant IDH1 R132H inhibitor with IC50 < 0.1 uM(A level in Patent).
Description

Mutant IDH1-IN-1 is a potent mutant IDH1 R132H inhibitor with IC50 < 0.1 uM(A level in Patent); more bioactivity information in Patent WO2012009678A1(Example 135).
Synonyms

Mutant IDH1-IN-1
Pathway

Metabolic Enzyme/Protease
Target

Dehydrogenase
Recptor

mutant IDH1 R132H
Research Area

Cancer
Indication

——

CAS Number

1355326-21-4
Formula Weight

498.59
Molecular Formula

C30H31FN4O2
Purity

>98%(HPLC)
Solubility

DMSO: 10 mM
SMILES

O=C(NC1CCCCC1)C(N(C(CN2C3=CC=CC=C3N=C2)=O)C4=CC=CC(F)=C4)C5=CC=CC=C5C
Chemical Name

2-(N-[2-(Benzimidazol-1-yl)acetyl]-3-fluoroanilino)-N-cyclohexyl-2-(2-methylphenyl)acetamide

1. Janeta Popovici-Muller, et al. Patent WO2012009678 A

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