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HhAntag
CAS No. 496794-70-8
HhAntag ( HhAntag; Hh-Antag; Hh Antag )
Catalog No. M17525 CAS No. 496794-70-8
HhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activity.
Purity : 96%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 102 | In Stock |
|
| 5MG | 185 | In Stock |
|
| 10MG | 320 | In Stock |
|
| 25MG | 529 | In Stock |
|
| 50MG | 771 | In Stock |
|
| 100MG | 1062 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameHhAntag
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NoteResearch use only, not for human use.
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Brief DescriptionHhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activity.
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DescriptionHhAntag is a GLI1-mediated transcription inhibitor. It acts as an inhibitor of the Shh pathway.
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SynonymsHhAntag; Hh-Antag; Hh Antag
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PathwayMembrane Transporter/Ion Channel
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TargetTRP/TRPV Channel
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RecptorGli
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number496794-70-8
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Formula Weight450.92
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Molecular FormulaC24H23ClN4O3
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Purity96%
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SolubilityDMSO : ≥ 100 mg/mL. 221.77 mM; H2O : < 0.1 mg/mL
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SMILESC(=O)(c1cc(cc(c1)OC)OC)Nc1cc(c(cc1)Cl)c1nc2c([nH]1)cc(cc2)N(C)C
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Chemical NameN-[4-Chloro-3-[6-(dimethylamino)-1H-benzimidazol-2-yl]phenyl]-3,5-dimethoxybenzamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Actis, Marcelo; Connelly, Michele C.; Mayasundari, Anand et al. Biopolymers (2011), 95(1), 24-30.
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