Gavestinel sodium( —— )

Catalog No. M33855 CAS No. 153436-38-5

Gavestinel (GV 150526) is a non-competitive NMDA receptor antagonist that is potent, selective and orally active.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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2MG	58	Get Quote
5MG	85	Get Quote
10MG	140	Get Quote
25MG	228	Get Quote
50MG	339	Get Quote
100MG	489	Get Quote
500MG	Get Quote	Get Quote
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Biological Information

Product Name

Gavestinel sodium
Note

Research use only, not for human use.
Brief Description

Gavestinel (GV 150526) is a non-competitive NMDA receptor antagonist that is potent, selective and orally active.
Description

Gavestinel (GV 150526A) is a potent, selective, orally active and non-competitive antagonist of NMDA receptor. Gavestinel binds to the glycine site of the NMDA receptor, with a pKi of 8.5. Gavestinel can be used for the research of acute ischemic stroke.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Membrane Transporter/Ion Channel
Target

iGluR
Recptor

iGluR | NMDAR
Research Area

——
Indication

——

Chemical Information

CAS Number

153436-38-5
Formula Weight

397.19
Molecular Formula

C18H11Cl2N2NaO3
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 100 mg/mL (251.77 mM; Ultrasonic )
SMILES

O=C(NC1=CC=CC=C1)/C=C/C2=C(C([O-])=O)NC3=CC(Cl)=CC(Cl)=C23.[Na+]
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Fabio RD, et, al. Substituted indole-2-carboxylates as in vivo potent antagonists acting as the strychnine-insensitive glycine binding site. J Med Chem. 1997 Mar 14;40(6):841-50.?

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