
GSK299115A
CAS No. 864082-35-9
GSK299115A( —— )
Catalog No. M34272 CAS No. 864082-35-9
GSK299115A (GSK-299115A) is a selective ROCK1 Inhibitor. GSK299115A exhibits IC50 of 8nM, 620nM, 560nM for ROCK1, RSK1, p70S6K, respectively.
Purity : >98% (HPLC)






Size | Price / USD | Stock | Quantity |
2MG | 511 | Get Quote |
![]() ![]() |
5MG | 772 | Get Quote |
![]() ![]() |
10MG | 1074 | Get Quote |
![]() ![]() |
25MG | 1546 | Get Quote |
![]() ![]() |
50MG | 2079 | Get Quote |
![]() ![]() |
100MG | 2673 | Get Quote |
![]() ![]() |
500MG | Get Quote | Get Quote |
![]() ![]() |
1G | Get Quote | Get Quote |
![]() ![]() |
Biological Information
-
Product NameGSK299115A
-
NoteResearch use only, not for human use.
-
Brief DescriptionGSK299115A (GSK-299115A) is a selective ROCK1 Inhibitor. GSK299115A exhibits IC50 of 8nM, 620nM, 560nM for ROCK1, RSK1, p70S6K, respectively.
-
DescriptionGSK299115A is a G Protein-coupled Receptor Kinase (GRK) and PKA inhibitor.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayOthers
-
TargetGRK (GPCRK)
-
RecptorGRK
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number864082-35-9
-
Formula Weight415.27
-
Molecular FormulaC20H16Cl2N4O2
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESC(NC=1C=C2C(=CC1)NN=C2)(=O)C=3C(CC(=O)NC3C)C4=CC(Cl)=C(Cl)C=C4
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Homan KT, et al. Identification and structure-function analysis of subfamily selective G protein-coupled receptor kinase inhibitors. ACS Chem Biol. 2015 Jan 16;10(1):310-9. ?
molnova catalog



related products
-
GSK-180736A
A highly selective and potent GRK2 inhibitor with IC50 of 0.77 uM.
-
GRK6-IN-1
GRK6-IN-1 (compound 18) is a potent inhibitor of G protein-coupled receptor kinase 6 (GRK6) with an IC50 of 120 nM, and has potential for study in multiple myeloma.
-
CCG-215022
CCG-215022 (CCG215022) is a potent and selective pan GRK inhibitor with IC50 of 0.15/0.38/3.9 uM for GRK2/5/1 respectively.