GR-64349 ( GR64349 )

Catalog No. M11556 CAS No. 137593-52-3

GR-64349 is a potent and selective tachykinin NK2 receptor agonist with EC50 of 3.7 nM.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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Biological Information

Product Name

GR-64349
Note

Research use only, not for human use.
Brief Description

GR-64349 is a potent and selective tachykinin NK2 receptor agonist with EC50 of 3.7 nM.
Description

GR-64349 is a potent and selective tachykinin NK2 receptor agonist with EC50 of 3.7 nM, displays >1000- and >300-fold selectivity over NK1 and NK3 receptors, respectively.Pain Discontinued
Synonyms

GR64349
Pathway

GPCR/G Protein
Target

Neurokinin Receptor
Recptor

Neurokinin Receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

137593-52-3
Formula Weight

921.12
Molecular Formula

C42H68N10O11S
Purity

>98% (HPLC)
Solubility

——
SMILES

CC(C)CC(C(=O)NC(CCSC)C(=O)N)N1CCC(C1=O)NC(=O)C(C(C)C)NC(=O)C(CC2=CC=CC=C2)NC(=O)C(CO)NC(=O)C(CC(=O)O)NC(=O)C(CCCCN)N
Chemical Name

KDSFVGLM (Modifications: Leu-7 = R-γ-lactam-Leu, Met-8 = C-terminal amide)

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Deal MJ, et al. J Med Chem. 1992 Oct 30;35(22):4195-204.
2. Chizh BA, et al. Br J Pharmacol. 1995 Jul;115(6):1013-9.
3. Chang Y, et al. J Pharmacol Exp Ther. 2000 Jul;294(1):147-54.

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