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GR-64349
CAS No. 137593-52-3
GR-64349 ( GR64349 )
Catalog No. M11556 CAS No. 137593-52-3
GR-64349 is a potent and selective tachykinin NK2 receptor agonist with EC50 of 3.7 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameGR-64349
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NoteResearch use only, not for human use.
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Brief DescriptionGR-64349 is a potent and selective tachykinin NK2 receptor agonist with EC50 of 3.7 nM.
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DescriptionGR-64349 is a potent and selective tachykinin NK2 receptor agonist with EC50 of 3.7 nM, displays >1000- and >300-fold selectivity over NK1 and NK3 receptors, respectively.Pain Discontinued
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SynonymsGR64349
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PathwayGPCR/G Protein
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TargetNeurokinin Receptor
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RecptorNeurokinin Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number137593-52-3
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Formula Weight921.12
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Molecular FormulaC42H68N10O11S
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Purity>98% (HPLC)
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Solubility——
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SMILESCC(C)CC(C(=O)NC(CCSC)C(=O)N)N1CCC(C1=O)NC(=O)C(C(C)C)NC(=O)C(CC2=CC=CC=C2)NC(=O)C(CO)NC(=O)C(CC(=O)O)NC(=O)C(CCCCN)N
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Chemical NameKDSFVGLM (Modifications: Leu-7 = R-γ-lactam-Leu, Met-8 = C-terminal amide)
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Deal MJ, et al. J Med Chem. 1992 Oct 30;35(22):4195-204.
2. Chizh BA, et al. Br J Pharmacol. 1995 Jul;115(6):1013-9.
3. Chang Y, et al. J Pharmacol Exp Ther. 2000 Jul;294(1):147-54.
2. Chizh BA, et al. Br J Pharmacol. 1995 Jul;115(6):1013-9.
3. Chang Y, et al. J Pharmacol Exp Ther. 2000 Jul;294(1):147-54.
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