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Home - Products - Metabolic Enzyme/Protease - Transferase - DGAT1-IN-1

DGAT1-IN-1

CAS No. 1449779-49-0

DGAT1-IN-1 ( —— )

Catalog No. M26665 CAS No. 1449779-49-0

DGAT1-IN-1 is a potent inhibitor of diacylglycerol O- acyltransferase type 1(DGAT1, IC50 of < 10 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    DGAT1-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    DGAT1-IN-1 is a potent inhibitor of diacylglycerol O- acyltransferase type 1(DGAT1, IC50 of < 10 nM).
  • Description
    DGAT1-IN-1 is a potent inhibitor of diacylglycerol O- acyltransferase type 1(DGAT1, IC50 of < 10 nM).(In Vitro):Various concentrations (0.0008 μΜ, 0.004 μΜ, 0.02 μΜ, 0.1 μΜ, 0.5 μΜ, 2.5 μΜ and 10.0 μΜ) of the compounds of Examples were added to individual wells prior to the addition of the cell lysates, or human or mouse liver microsomes.
  • Synonyms
    ——
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Transferase
  • Recptor
    Centromere-Associated Protein E
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1449779-49-0
  • Formula Weight
    551.6
  • Molecular Formula
    C30H28F3N3O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    OC(=O)C[C@H]1CC[C@@H](CC1)c1ccc(cc1)-c1ccc2nc(cn2c1)C(=O)NCc1ccc(OC(F)(F)F)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Qian X, et al. Discovery of the First Potent and Selective Inhibitor of Centromere-Associated Protein E: GSK923295. ACS Med Chem Lett. 2010 Jan 19;1(1):30-4.
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