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DDR2-IN-5
CAS No. 1796592-06-7
DDR2-IN-5( —— )
Catalog No. M12712 CAS No. 1796592-06-7
DDR2-IN-5 is a potent, dual DDR2/SRC inhibitor with IC50 of 56/12 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameDDR2-IN-5
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NoteResearch use only, not for human use.
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Brief DescriptionDDR2-IN-5 is a potent, dual DDR2/SRC inhibitor with IC50 of 56/12 nM.
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DescriptionDDR2-IN-5 is a potent, dual DDR2/SRC inhibitor with IC50 of 56/12 nM, potently suppresses DDR2 mutated cell lines HCC-366 and NCI-H2286 with IC50 of 0.44 uM and 0.29 uM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayTyrosine Kinase
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TargetDDR
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RecptorDDR
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Research Area——
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Indication——
Chemical Information
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CAS Number1796592-06-7
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Formula Weight605.666
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Molecular FormulaC32H34F3N7O2
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical NameN-(5-((4-((4-ethylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)carbamoyl)-2-methylphenyl)-5-(1-methyl-1H-pyrazol-4-yl)nicotinamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Terai H, et al. ACS Chem Biol. 2015 Dec 18;10(12):2687-96.
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DDR2-IN-5
DDR2-IN-5 is a potent, dual DDR2/SRC inhibitor with IC50 of 56/12 nM.
