Cart
sales@molnova.com
Home - Products - GPCR/G Protein - Antibacterial - Contezolid

Contezolid

CAS No. 1112968-42-9

Contezolid ( MRX I )

Catalog No. M10415 CAS No. 1112968-42-9

Contezolid (MRX I) is an orally active oxazolidinone agent with antibacterial activity Gram-positive pathogens, including MRSA, penicillin-PRSP, PISP, and vancomycin-resistant enterococci (VRE) with MIC of 0.25-4 ug/mL.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 598 Get Quote
50MG 2502 Get Quote
100MG 3330 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote
Group Booking Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    Contezolid
  • Note
    Research use only, not for human use.
  • Brief Description
    Contezolid (MRX I) is an orally active oxazolidinone agent with antibacterial activity Gram-positive pathogens, including MRSA, penicillin-PRSP, PISP, and vancomycin-resistant enterococci (VRE) with MIC of 0.25-4 ug/mL.
  • Description
    Contezolid (MRX I) is an orally active oxazolidinone agent with antibacterial activity Gram-positive pathogens, including MRSA, penicillin-PRSP, PISP, and vancomycin-resistant enterococci (VRE) with MIC of 0.25-4 ug/mL; demonstrates the same or better efficacy than linezolid in both systemic and local infection models against the tested strains.Bacterial Infection Phase 3 Clinical
  • Synonyms
    MRX I
  • Pathway
    GPCR/G Protein
  • Target
    Antibacterial
  • Recptor
    Antibacterial
  • Research Area
    Infection
  • Indication
    Bacterial Infection

Chemical Information

  • CAS Number
    1112968-42-9
  • Formula Weight
    408.34
  • Molecular Formula
    C18H15F3N4O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C1CCN(C2=C(F)C=C(N3C(O[C@@H](CNC4=NOC=C4)C3)=O)C(F)=C2F)C=C1
  • Chemical Name
    1-{2,3,6-trifluoro-4-[(5S)-5-{[(1,2-oxazol-3-yl)amino]methyl}-2-oxo-1,3-oxazolidin-3-yl]phenyl}-2,3-dihydropyridin-4(1H)-one

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Li CR, et al. Antimicrob Agents Chemother. 2014;58(4):2418-21.
2. Gordeev MF, et al. J Med Chem. 2014 Jun 12;57(11):4487-97.
3. Meng J, et al. Drug Metab Dispos. 2015 May;43(5):646-59.
4. Eckburg PB, et al. Antimicrob Agents Chemother. 2017 Mar 24;61(4). pii: e02181-16.
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • QcrB inhibitor TB47

    QcrB inhibitor TB47 (TB47) is a novel antimycobacterial agent that fuctions as a putative respiratory complex III (QcrB) inhibitor with MIC of 0.016-0.5 ug/mL against a panel of 56 M.

  • 6-Diazo-5-oxo-L-nor-...

    L-6-Diazo-5-oxonorleucine is an antagonist of glutaminases (Ki : 6 μM). It is an antineoplastic antibiotic produced by an unidentified species of Streptomyces from Peruvian soil.

  • Methicillin sodium

    Methicillin Sodium is the sodium salt form of methicillin a semisynthetic beta-lactam penicillin antibiotic with beta-lactamase resistant activity.

Sign In Join Free