Cetrorelix
CAS No. 145672-81-7
Cetrorelix( —— )
Catalog No. M20166 CAS No. 145672-81-7
Cetrorelix Acetate is gonadotropin-releasing hormone?(GnRH)?receptor antagonist with an?IC50?of 1.21 nM.
Purity : >98% (HPLC)
Size | Price / USD | Stock | Quantity |
2MG | 61 | In Stock |
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5MG | 86 | In Stock |
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10MG | 146 | In Stock |
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25MG | 304 | In Stock |
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50MG | 501 | In Stock |
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100MG | 713 | In Stock |
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200MG | Get Quote | In Stock |
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500MG | Get Quote | In Stock |
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1G | Get Quote | In Stock |
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Biological Information
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Product NameCetrorelix
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NoteResearch use only, not for human use.
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Brief DescriptionCetrorelix Acetate is gonadotropin-releasing hormone?(GnRH)?receptor antagonist with an?IC50?of 1.21 nM.
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DescriptionCetrorelix Acetate is gonadotropin-releasing hormone?(GnRH)?receptor antagonist with an?IC50?of 1.21 nM.(In Vitro):Cetrorelix Acetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix Acetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells.
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In VitroCetrorelix Acetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix Acetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells.
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorGNRHR
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Research AreaOthers
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Indication——
Chemical Information
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CAS Number145672-81-7
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Formula Weight1491.11
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Molecular FormulaC70H92ClN17O14.C2H4O2
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Purity>98% (HPLC)
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SolubilityDMSO:50 mg/mL?(33.53 mM)
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SMILESCC(O)=O.CC(C)C[C@H](NC(=O)[C@@H](CCCNC(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CO)NC(=O)[C@@H](Cc1cccnc1)NC(=O)[C@@H](Cc1ccc(Cl)cc1)NC(=O)[C@@H](Cc1ccc2ccccc2c1)NC(C)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N1CCC[C@H]1C(=O)N[C@H](C)C(N)=O
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Chemical Name(S)-1-(((R)-2-((S)-2-((S)-2-((R)-2-((R)-2-((R)-2-acetamido-3-(naphthalen-2-yl)propanamido)-3-(4-chlorophenyl)propanamido)-3-(pyridin-3-yl)propanamido)-3-hydroxypropanamido)-3-(4-hydroxyphenyl)propanamido)-5-ureidopentanoyl)-L-leucyl-L-arginyl)-N-((R)-1-amino-1-oxopropan-2-yl)pyrrolidine-2-carboxamide acetate
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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