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CDK9-PROTAC
CAS No. 2118356-96-8
CDK9-PROTAC ( CDK9PROTAC; CDK9 PROTAC; CDK9-PROTAC )
Catalog No. M13368 CAS No. 2118356-96-8
CDK9-PROTAC is a heterobifunctional small molecule PROTAC capable of cereblon mediated proteasomal degradation of CDK9.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 298 | In Stock |
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| 10MG | 478 | In Stock |
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| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameCDK9-PROTAC
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NoteResearch use only, not for human use.
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Brief DescriptionCDK9-PROTAC is a heterobifunctional small molecule PROTAC capable of cereblon mediated proteasomal degradation of CDK9.
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DescriptionCDK9-PROTAC is a heterobifunctional small molecule PROTAC capable of cereblon mediated proteasomal degradation of CDK9; selectively degrades CDK9 while sparing other CDK family members in HCT116 cells.
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SynonymsCDK9PROTAC; CDK9 PROTAC; CDK9-PROTAC
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PathwayPROTACs
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TargetPROTAC
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RecptorPROTAC
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Research Area——
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Indication——
Chemical Information
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CAS Number2118356-96-8
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Formula Weight613.67
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Molecular FormulaC33H35N5O7
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Purity>98% (HPLC)
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SolubilityDMSO : ≥ 104 mg/mL 169.47 mM
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SMILESO=C(NC1=NNC(C2CCC2)=C1)CC3=CC=C(OCCCCCOC4=CC=CC(C(N5C(CC6)C(NC6=O)=O)=O)=C4C5=O)C=C3
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Chemical NameN-(5-cyclobutyl-1H-pyrazol-3-yl)-2-(4-((5-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)pentyl)oxy)phenyl)acetamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Robb CM, et al. Chem Commun (Camb). 2017 Jul 4;53(54):7577-7580.
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