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C646
CAS No. 328968-36-1
C646 ( C646; C-646; C 646 )
Catalog No. M14079 CAS No. 328968-36-1
C646 is an inhibitor for histone acetyltransferase, and inhibits p300 with a Ki of 400 nM in a cell-free assay.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 37 | In Stock |
|
| 5MG | 57 | In Stock |
|
| 10MG | 88 | In Stock |
|
| 25MG | 185 | In Stock |
|
| 50MG | 360 | In Stock |
|
| 100MG | 533 | In Stock |
|
| 500MG | 1143 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameC646
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NoteResearch use only, not for human use.
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Brief DescriptionC646 is an inhibitor for histone acetyltransferase, and inhibits p300 with a Ki of 400 nM in a cell-free assay.
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DescriptionC646 is an inhibitor for histone acetyltransferase, and inhibits p300 with a Ki of 400 nM in a cell-free assay. Preferentially selective for p300 versus other acetyltransferases.
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SynonymsC646; C-646; C 646
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PathwayChromatin/Epigenetic
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TargetEpigenetic Reader Domain
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Recptorp300/CBP
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Research AreaOther Indications
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Indication——
Chemical Information
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CAS Number328968-36-1
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Formula Weight445.42
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Molecular FormulaC24H19N3O6
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Purity>98%(HPLC)
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SolubilityDMSO: 13 mg/mL (29.18 mM)
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SMILESO=C(O)C1=CC=C(N2N=C(C)/C(C2=O)=C\C3=CC=C(C4=CC(C)=C(C)C=C4[N+]([O-])=O)O3)C=C1
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Chemical Name(E)-4-(4-((5-(4,5-dimethyl-2-nitrophenyl)furan-2-yl)methylene)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl)benzoic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Bowers EM, et al. Chem Biol, 2010, 17(5), 471-482.
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