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BRD9539
CAS No. 1374601-41-8
BRD9539 ( —— )
Catalog No. M20714 CAS No. 1374601-41-8
BRD9539 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2) also known as G9a with an IC50 value of 6.3 μM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 27 | In Stock |
|
| 5MG | 42 | In Stock |
|
| 10MG | 71 | In Stock |
|
| 25MG | 119 | In Stock |
|
| 50MG | 176 | In Stock |
|
| 100MG | 259 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBRD9539
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NoteResearch use only not for human use.
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Brief DescriptionBRD9539 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2) also known as G9a with an IC50 value of 6.3 μM.
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DescriptionBRD9539 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2) also known as G9a with an IC50 value of 6.3 μM.
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetHistone Demethylase
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RecptorG9a
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Research Area——
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Indication——
Chemical Information
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CAS Number1374601-41-8
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Formula Weight399.44
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Molecular FormulaC24H21N3O3
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Purity>98% (HPLC)
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SolubilityDMSO:35 mg/mL (87.62 mM)
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SMILESOC(=O)c1ccc2n(CCCc3ccccc3)c(NC(=O)c3ccccc3)nc2c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Yuan Y Wang Q Paulk J et al. A Small-Molecule Probe of the Histone Methyltransferase G9a Induces Cellular Senescence in Pancreatic Adenocarcinoma[J]. ACS Chemical Biology 2012 7(7):1152-1157.
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