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BRD2492
CAS No. 1821669-43-5
BRD2492( BRD 2492 )
Catalog No. M12810 CAS No. 1821669-43-5
BRD2492 is a highly potent, selective HDAC1/2 inhibitor (IC50=2/19 nM, respectively).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameBRD2492
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NoteResearch use only, not for human use.
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Brief DescriptionBRD2492 is a highly potent, selective HDAC1/2 inhibitor (IC50=2/19 nM, respectively).
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DescriptionBRD2492 is a highly potent, selective HDAC1/2 inhibitor (IC50=2/19 nM, respectively) that displays excellent selectivity versus HDAC3 (IC50=2.08 uM, ≥110-fold selectivity) and all other HDAC isoforms, increases caspase-3 activation.
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In Vitro——
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In Vivo——
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SynonymsBRD 2492
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PathwayCell Cycle/DNA Damage
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TargetHDAC
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RecptorHDAC
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Research Area——
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Indication——
Chemical Information
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CAS Number1821669-43-5
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Formula Weight346.39
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Molecular FormulaC20H18N4O2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 31.25 mg/mL (90.22 mM)
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SMILESO=C(NC1=CC(C2=CC=NC=C2)=CC=C1N)C3=CC=C(NC(C)=O)C=C3
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Chemical Name4-Acetylamino-N-(2-amino-5-pyridin-4-yl-phenyl)-benzamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Wagner FF, et al. ACS Chem Biol. 2016 Feb 19;11(2):363-74.
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