Cart
sales@molnova.com
BMS-193885
CAS No. 186185-03-5
BMS-193885 ( —— )
Catalog No. M26631 CAS No. 186185-03-5
BMS-193885 is a potent, selective, competitive, and brain penetrant neuropeptide Y1 receptor antagonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 110 | Get Quote |
|
| 10MG | 177 | Get Quote |
|
| 25MG | 357 | Get Quote |
|
| 50MG | 530 | Get Quote |
|
| 100MG | 759 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameBMS-193885
-
NoteResearch use only, not for human use.
-
Brief DescriptionBMS-193885 is a potent, selective, competitive, and brain penetrant neuropeptide Y1 receptor antagonist.
-
DescriptionBMS-193885 is a potent, selective, competitive, and brain penetrant neuropeptide Y1 receptor antagonist. With a Ki of 3.3 nM, and has an IC50 of 5.9 nM for hY1. It displays > 100, > 160, > 160 and > 160-fold selectivity over α1, hY2, hY4 and hY5 receptors, respectively.
-
Synonyms——
-
PathwayOthers
-
TargetOther Targets
-
Recptor——
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number186185-03-5
-
Formula Weight590.7
-
Molecular FormulaC33H42N4O6
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESCOC(=O)C1=C(C)NC(C)=C(C1c1cccc(NC(=O)NCCCN2CCC(CC2)c2cccc(OC)c2)c1)C(=O)OC
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Kutluay VM, et al. Cytotoxic phenylethanoid glycosides from Digitalis davisiana Heywood: Evaluation of structure activity relationships and chemotaxonomical significance of isolated compounds. Fitoterapia. 2019 Jun;135:90-98.
molnova catalog
related products
-
Dichlorodiphenylmeth...
Used as pharmaceutical intermediates.
-
TK216
TK216 is a potent inhibitor of E26 transformation-specific (ETS) with anticancer activity.In DLBCL cell lines, TK216 (500 nM; for 24-72 hours) induces apoptosis.
-
Plantagoside
Plantagoside is a specific non-competitive inhibitor for jack bean alpha-mannosidase (IC50: 5 μM). It also is a potent inhibitor of the Maillard reaction.
