BMS-193885
CAS No. 186185-03-5
BMS-193885 ( —— )
Catalog No. M26631 CAS No. 186185-03-5
BMS-193885 is a potent, selective, competitive, and brain penetrant neuropeptide Y1 receptor antagonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 110 | Get Quote |
|
10MG | 177 | Get Quote |
|
25MG | 357 | Get Quote |
|
50MG | 530 | Get Quote |
|
100MG | 759 | Get Quote |
|
200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
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Product NameBMS-193885
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NoteResearch use only, not for human use.
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Brief DescriptionBMS-193885 is a potent, selective, competitive, and brain penetrant neuropeptide Y1 receptor antagonist.
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DescriptionBMS-193885 is a potent, selective, competitive, and brain penetrant neuropeptide Y1 receptor antagonist. With a Ki of 3.3 nM, and has an IC50 of 5.9 nM for hY1. It displays > 100, > 160, > 160 and > 160-fold selectivity over α1, hY2, hY4 and hY5 receptors, respectively.
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Synonyms——
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PathwayOthers
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TargetOther Targets
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number186185-03-5
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Formula Weight590.7
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Molecular FormulaC33H42N4O6
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Purity>98% (HPLC)
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Solubility——
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SMILESCOC(=O)C1=C(C)NC(C)=C(C1c1cccc(NC(=O)NCCCN2CCC(CC2)c2cccc(OC)c2)c1)C(=O)OC
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Kutluay VM, et al. Cytotoxic phenylethanoid glycosides from Digitalis davisiana Heywood: Evaluation of structure activity relationships and chemotaxonomical significance of isolated compounds. Fitoterapia. 2019 Jun;135:90-98.
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