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Avanafil
CAS No. 330784-47-9
Avanafil ( TA1790;TA 1790;TA-1790 )
Catalog No. M14101 CAS No. 330784-47-9
A potent and highly selective PDE5 inhibitor (IC50=5.2 nM) for erectile dysfunction.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 25MG | 42 | In Stock |
|
| 50MG | 52 | In Stock |
|
| 100MG | 85 | In Stock |
|
| 200MG | 102 | In Stock |
|
| 500MG | 125 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameAvanafil
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NoteResearch use only, not for human use.
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Brief DescriptionA potent and highly selective PDE5 inhibitor (IC50=5.2 nM) for erectile dysfunction.
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DescriptionA potent and highly selective PDE5 inhibitor (IC50=5.2 nM) for erectile dysfunction; shows no significant effect on PDE1, PDE6 and PDE11.Sexual Dysfunction Approved
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SynonymsTA1790;TA 1790;TA-1790
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PathwayAngiogenesis
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TargetPDE
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RecptorPDE5
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Research AreaEndocrinology
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IndicationSexual Dysfunction
Chemical Information
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CAS Number330784-47-9
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Formula Weight483.95
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Molecular FormulaC23H26ClN7O3
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESO=C(C1=CN=C(N2[C@H](CO)CCC2)N=C1NCC3=CC=C(OC)C(Cl)=C3)NCC4=NC=CC=N4
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Chemical Name5-Pyrimidinecarboxamide, 4-[[(3-chloro-4-methoxyphenyl)methyl]amino]-2-[(2S)-2-(hydroxymethyl)-1-pyrrolidinyl]-N-(2-pyrimidinylmethyl)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kotera J, et al. J Urol. 2012 Aug;188(2):668-74.
2. Limin M, et al. Expert Opin Investig Drugs. 2010 Nov;19(11):1427-37.
3. Wang R, et al. J Sex Med. 2012 Aug;9(8):2122-9.
2. Limin M, et al. Expert Opin Investig Drugs. 2010 Nov;19(11):1427-37.
3. Wang R, et al. J Sex Med. 2012 Aug;9(8):2122-9.
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