
AZD-9567
CAS No. 1893415-00-3
AZD-9567( AZD9567 )
Catalog No. M12972 CAS No. 1893415-00-3
AZD-9567 (AZD9567) is a potent, selective, non-steroidal and orally available selective glucocorticoid receptor modulator (SGRM) for treatment of rheumatoid arthritis.
Purity : >98% (HPLC)






Size | Price / USD | Stock | Quantity |
5MG | 484 | Get Quote |
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10MG | 699 | Get Quote |
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25MG | 1062 | Get Quote |
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50MG | 1431 | Get Quote |
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100MG | 1917 | Get Quote |
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200MG | Get Quote | Get Quote |
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500MG | Get Quote | Get Quote |
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1G | Get Quote | Get Quote |
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Biological Information
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Product NameAZD-9567
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NoteResearch use only, not for human use.
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Brief DescriptionAZD-9567 (AZD9567) is a potent, selective, non-steroidal and orally available selective glucocorticoid receptor modulator (SGRM) for treatment of rheumatoid arthritis.
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DescriptionAZD-9567 (AZD9567) is a potent, selective, non-steroidal and orally available selective glucocorticoid receptor modulator (SGRM) for treatment of rheumatoid arthritis.Rheumatoid Arthritis Phase 2 Clinical.
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In Vitro——
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In VivoMizacorat (15 mg/kg/day, Oral gavage daily for 8 days) treatment shows excellent in vivo efficacy in a rat model of joint inflammation. Animal Model:Antigen-induced joint inflammation model in female Lewis rats (175-200 g), sensitized by an intra-articular injection of 5 μg of SCW.Dosage:15 mg/kg/day.Administration:Oral gavage daily for 8 days.Result:Inhibited ankle swelling in the rat SCW model.
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SynonymsAZD9567
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PathwayEndocrinology/Hormones
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TargetGR
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RecptorGR
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Research AreaInflammation/Immunology
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IndicationRheumatoid Arthritis
Chemical Information
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CAS Number1893415-00-3
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Formula Weight494.533
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Molecular FormulaC27H28F2N4O3
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESCC(F)(F)C(N[C@@H](C(C)C)[C@H](OC1=CC2=C(N(C(C=C3)=CN(C)C3=O)N=C2)C=C1)C4=CC=CC=C4)=O
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Chemical Name2,2-Difluoro-N-[(1R,2S)-3-methyl-1-[[1-(1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-1H-indazol-5-yl]oxy]-1-phenylbutan-2-yl]propanamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ripa L, et al. J Med Chem. 2018 Mar 8;61(5):1785-1799.
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