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ASP4132
CAS No. 1640294-30-9
ASP4132 ( —— )
Catalog No. M22042 CAS No. 1640294-30-9
ASP4132 is an orally active AMPK activator (EC50 : 18 nM), has anti-cancer activity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 79 | Get Quote |
|
| 5MG | 120 | Get Quote |
|
| 10MG | 186 | Get Quote |
|
| 25MG | 338 | Get Quote |
|
| 50MG | 507 | Get Quote |
|
| 100MG | 714 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameASP4132
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NoteResearch use only, not for human use.
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Brief DescriptionASP4132 is an orally active AMPK activator (EC50 : 18 nM), has anti-cancer activity.
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DescriptionASP4132 is an orally active AMPK activator (EC50 : 18 nM), has anti-cancer activity.
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetAMPK
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RecptorAMPK
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Research Area——
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Indication——
Chemical Information
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CAS Number1640294-30-9
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Formula Weight937.06
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Molecular FormulaC46H51F3N6O8S2
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Purity>98% (HPLC)
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SolubilityDMSO:230 mg/mL (245.45 mM; Need ultrasonic); Methanol:8.33 mg/mL (8.89 mM; Need ultrasonic)
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SMILESCC1=CC=C(C=C1)S(O)(=O)=O.CC1=CC=C(C=C1)S(O)(=O)=O.COC1=CC=C(CN2CCC(CC2)C2=CC=C3N=C(NC3=C2)C(=O)N2CCN(CC3=CC=C(C=C3)C(F)(F)F)CC2)C=N1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kazuyuki Kuramoto , Yuki Sawada, Tomohiro Yamada,et al.Novel Indirect AMP-Activated Protein Kinase Activators: Identification of a Second-Generation Clinical Candidate with Improved Physicochemical Properties and Reduced hERG Inhibitory Activity.Chem Pharm Bull (Tokyo). 2020;68(5):452-465.
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