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ARV-110
CAS No. 2222112-77-6
ARV-110 ( —— )
Catalog No. M24006 CAS No. 2222112-77-6
ARV-110 is an oral degrader of androgen receptor PROTAC for prostate cancer treatment.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 77 | In Stock |
|
| 5MG | 125 | In Stock |
|
| 10MG | 194 | In Stock |
|
| 25MG | 382 | In Stock |
|
| 50MG | 491 | In Stock |
|
| 100MG | 707 | In Stock |
|
| 200MG | 981 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameARV-110
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NoteResearch use only, not for human use.
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Brief DescriptionARV-110 is an oral degrader of androgen receptor PROTAC for prostate cancer treatment.
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DescriptionARV-110 is an oral degrader of androgen receptor PROTAC for prostate cancer treatment.
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetAndrogen Receptor (AR)
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RecptorAndrogen Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number2222112-77-6
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Formula Weight812.3
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Molecular FormulaC41H43ClFN9O6
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Purity>98% (HPLC)
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SolubilityDMSO:46 mg/mL (56.63 mM; Need ultrasonic)
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SMILESClC1=CC(O[C@H]2CC[C@@H](CC2)NC(C3=CC=C(N=N3)N4CCC(CC4)CN5CCN(CC5)C6=CC(C(N7C8CCC(NC8=O)=O)=O)=C(C=C6F)C7=O)=O)=CC=C1C#N
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Taavi K Neklesa,et al. ARV-110: an oral androgen receptor PROTAC degrader for prostate cancer. GU ASCO 2019
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