ABBV-744
CAS No. 2138861-99-9
ABBV-744 ( ABBV744 )
Catalog No. M13413 CAS No. 2138861-99-9
ABBV-744 (ABBV744) is a potent, BDII-selective BET bromodomain inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 49 | In Stock |
|
5MG | 87 | In Stock |
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10MG | 138 | In Stock |
|
25MG | 284 | In Stock |
|
50MG | 410 | In Stock |
|
100MG | 500 | In Stock |
|
200MG | 718 | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
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Product NameABBV-744
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NoteResearch use only, not for human use.
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Brief DescriptionABBV-744 (ABBV744) is a potent, BDII-selective BET bromodomain inhibitor.
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DescriptionABBV-744 (ABBV744) is a potent, BDII-selective BET bromodomain inhibitor, ABBV-744 is a potent, selective inhibitor of the AR transcription activity; induces tumor growth inhibition in LNCaP and MDA-Pca-2b xenograft models.Prostate Cancer Phase 1 Clinical
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SynonymsABBV744
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PathwayChromatin/Epigenetic
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TargetBromodomain
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RecptorBET bromodomain
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Research AreaCancer
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IndicationProstate Cancer
Chemical Information
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CAS Number2138861-99-9
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Formula Weight491.56
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Molecular FormulaC28H30FN3O4
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Purity>98% (HPLC)
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SolubilityDMSO: 10 mM ( < 1 mg/ml refers to the product slightly soluble or insoluble )
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SMILESO=C(C(N1)=CC(C(C2=CC(C(C)(O)C)=CC=C2OC3=C(C)C=C(F)C=C3C)=CN4C)=C1C4=O)NCC
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Chemical Name1H-Pyrrolo[2,3-c]pyridine-2-carboxamide, N-ethyl-4-[2-(4-fluoro-2,6-dimethylphenoxy)-5-(1-hydroxy-1-methylethyl)phenyl]-6,7-dihydro-6-methyl-7-oxo-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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