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GSK525768A
CAS No. 1260530-25-3
GSK525768A ( GSK 525768A;GSK-525768A )
Catalog No. M11076 CAS No. 1260530-25-3
GSK525768A is an enantiomer, negative control compound of I-BET762 (GSK525762A).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 312 | Get Quote |
|
| 50MG | 1377 | Get Quote |
|
| 100MG | 1791 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameGSK525768A
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NoteResearch use only, not for human use.
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Brief DescriptionGSK525768A is an enantiomer, negative control compound of I-BET762 (GSK525762A).
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DescriptionGSK525768A is an enantiomer, negative control compound of I-BET762 (GSK525762A), shows no activity against BET family proteins BRD2, BRD3 and BRD4.
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SynonymsGSK 525768A;GSK-525768A
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PathwayChromatin/Epigenetic
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TargetBromodomain
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RecptorBromodomain
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Research AreaInflammation/Immunology
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Indication——
Chemical Information
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CAS Number1260530-25-3
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Formula Weight423.90
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Molecular FormulaC22H22ClN5O2
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESCCNC(=O)CC1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C
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Chemical Name4H-[1,2,4]Triazolo[4,3-a][1,4]benzodiazepine-4-acetamide, 6-(4-chlorophenyl)-N-ethyl-8-methoxy-1-methyl-, (4R)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Nicodeme E, et al. Nature. 2010 Dec 23;468(7327):1119-23.
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